Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 7947
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225264(3-Bromo-N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d]...)
Affinity DataIC50: 1.32E+3nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225261(2-Methoxy-N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[...)
Affinity DataIC50: 1.75E+3nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225253(2-Methoxy-N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[...)
Affinity DataIC50: 2.63E+3nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225263(Brd4470)
Affinity DataIC50: 6.10E+3nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225260(2-Fluoro-N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d...)
Affinity DataIC50: 9.59E+3nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225262(N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d]imidazol...)
Affinity DataIC50: 1.22E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225249(2-Methoxy-N-(2-phenylbenzo[d]oxazol-6-yl)benzamide...)
Affinity DataIC50: 1.28E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225242(ErbB2-pep | 2-Methoxy-N-(2-phenylbenzo[d]oxazol-6-...)
Affinity DataIC50: 1.53E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225251(3-Bromo-N-(2-phenylbenzo[d]oxazol-6-yl)benzamide (...)
Affinity DataIC50: 1.53E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225254(N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d]imidazol...)
Affinity DataIC50: 1.60E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225256(4-Fluoro-N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d...)
Affinity DataIC50: 1.61E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225259(4-(tert-Butyl)-N-(2-phenyl-1-(3-phenylpropyl)-1H-b...)
Affinity DataIC50: 1.63E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225257(4-Cyano-N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d]...)
Affinity DataIC50: 1.88E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225244(IGF1R-pep | N-(2-phenylbenzo[d]oxazol-6-yl)-4-(tri...)
Affinity DataIC50: 1.90E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225258(2-Bromo-N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d]...)
Affinity DataIC50: 2.08E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225255(N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d]imidazol...)
Affinity DataIC50: 2.19E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225243(IR-pep | N-(2-Phenyl-1H-1l3-benzo[d]oxazol-6-yl)-4...)
Affinity DataIC50: 2.62E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225246(4-Cyano-N-(2-phenylbenzo[d]oxazol-6-yl)benzenesulf...)
Affinity DataIC50: 3.04E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225240(PLCγ1-pep | 3,5-Difluoro-N-(2-phenylbenzo[d]o...)
Affinity DataIC50: 3.32E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225252(3-Nitro-N-(2-phenyl-1-(3-phenylpropyl)-1H-benzo[d]...)
Affinity DataIC50: 3.54E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225248(4-(tert-Butyl)-N-(2-phenylbenzo[d]oxazol-6-yl)benz...)
Affinity DataIC50: 3.63E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225241(MT-pep | 3-Nitro-N-(2-phenylbenzo[d]oxazol-6-yl)be...)
Affinity DataIC50: 4.00E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225250(2-Fluoro-N-(2-phenylbenzo[d]oxazol-6-yl)benzamide ...)
Affinity DataIC50: 4.00E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225247(2-Bromo-N-(2-phenylbenzo[d]oxazol-6-yl)benzenesulf...)
Affinity DataIC50: 4.00E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225245(IRS2-pep | 4-Fluoro-N-(2-phenylbenzo[d]oxazol-6-yl...)
Affinity DataIC50: 4.00E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed