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Found 34 Enz. Inhib. hit(s) with all data for entry = 50001032
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268048(CHEMBL4098491)
Affinity DataKi:  3.19E+3nMAssay Description:Mixed-type inhibition of electric eel AChE using varying levels of acetylthiocholine iodide as substrate measured for 2 mins by Lineweaver-Burk plot ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM16047((4S)-4-[(2S)-2-[(2R,4S,5S)-5-[(2S)-2-[(2S)-2-[(4S)...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human BACE1 using Rh-EVNLDAEFK-quencher as substrate measured after 60 mins by FRET assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  31nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM10949(3-(4-{[Benzyl(methyl)amino]methyl}-phenyl)-6,7-dim...)
Affinity DataIC50:  45nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50362874(CHEMBL1940735)
Affinity DataIC50:  360nMAssay Description:Inhibition of AChE in Sprague-Dawley rat brain homogenates using [3H]-acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268048(CHEMBL4098491)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268060(CHEMBL4077242)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268040(CHEMBL4104739)
Affinity DataIC50:  2.05E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268043(CHEMBL4067112)
Affinity DataIC50:  3.25E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268061(CHEMBL4068753)
Affinity DataIC50:  6.33E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  8.73E+3nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268049(CHEMBL4060097)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268045(CHEMBL4078051)
Affinity DataIC50:  1.46E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268039(CHEMBL4072501)
Affinity DataIC50:  2.39E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268041(CHEMBL4086849)
Affinity DataIC50:  2.56E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268059(CHEMBL4103820)
Affinity DataIC50:  3.14E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268058(CHEMBL4080474)
Affinity DataIC50:  3.29E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268043(CHEMBL4067112)
Affinity DataIC50:  3.42E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268048(CHEMBL4098491)
Affinity DataIC50:  4.57E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268049(CHEMBL4060097)
Affinity DataIC50:  5.23E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268060(CHEMBL4077242)
Affinity DataIC50:  5.82E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268040(CHEMBL4104739)
Affinity DataIC50:  6.38E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268039(CHEMBL4072501)
Affinity DataIC50:  8.84E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268061(CHEMBL4068753)
Affinity DataIC50:  8.92E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268045(CHEMBL4078051)
Affinity DataIC50:  9.15E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268041(CHEMBL4086849)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268059(CHEMBL4103820)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268058(CHEMBL4080474)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268046(CHEMBL4102317)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268044(CHEMBL4094574)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268046(CHEMBL4102317)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268047(CHEMBL4076497)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268044(CHEMBL4094574)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50268047(CHEMBL4076497)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured for 6 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed