Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50002543
TargetAndrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459874BDBM50459874(CHEMBL4226259)
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459869BDBM50459869(CHEMBL4227715)
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459873BDBM50459873(CHEMBL4225186)
Affinity DataIC50: 27nMAssay Description:Displacement of [17-alpha-methyl-H-3] mibolerone from wild-type androgen receptor (unknown origin) expressed in human Freestyle293F cells measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459875BDBM50459875(CHEMBL4226844)
Affinity DataIC50: 53nMAssay Description:Binding affinity to androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459868BDBM50459868(CHEMBL4225339)
Affinity DataIC50: 54nMAssay Description:Binding affinity to androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459871BDBM50459871(CHEMBL4226314)
Affinity DataIC50: 190nMAssay Description:Displacement of [17-alpha-methyl-H-3] mibolerone from wild-type androgen receptor (unknown origin) expressed in human Freestyle293F cells measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459866BDBM50459866(CHEMBL4226899)
Affinity DataIC50: 190nMAssay Description:Displacement of [17-alpha-methyl-H-3] mibolerone from wild-type androgen receptor (unknown origin) expressed in human Freestyle293F cells measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459870BDBM50459870(CHEMBL4227287)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [17-alpha-methyl-H-3] mibolerone from wild-type androgen receptor (unknown origin) expressed in human Freestyle293F cells measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459867BDBM50459867(CHEMBL4226575)
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity to androgen receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459872BDBM50459872(CHEMBL4227353)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [17-alpha-methyl-H-3] mibolerone from wild-type androgen receptor (unknown origin) expressed in human Freestyle293F cells measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed