Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50000576
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254131(CHEMBL4094845)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254132(CHEMBL4083940)
Affinity DataKi:  0.211nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254124(CHEMBL4103044)
Affinity DataKi:  0.221nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254124(CHEMBL4103044)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at human recombinant DOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254133(CHEMBL4076632)
Affinity DataKi:  0.265nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254133(CHEMBL4076632)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254132(CHEMBL4083940)
Affinity DataEC50:  0.310nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254124(CHEMBL4103044)
Affinity DataKi:  0.313nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254133(CHEMBL4076632)
Affinity DataKi:  0.336nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254123(CHEMBL4068691)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity at human recombinant DOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254131(CHEMBL4094845)
Affinity DataKi:  0.356nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254132(CHEMBL4083940)
Affinity DataKi:  0.362nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254130(CHEMBL4061334)
Affinity DataEC50:  0.420nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254131(CHEMBL4094845)
Affinity DataEC50:  0.430nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254124(CHEMBL4103044)
Affinity DataKi:  0.455nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254123(CHEMBL4068691)
Affinity DataKi:  0.458nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254131(CHEMBL4094845)
Affinity DataKi:  0.479nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254120(CHEMBL4076681)
Affinity DataKi:  0.522nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254133(CHEMBL4076632)
Affinity DataKi:  0.545nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254123(CHEMBL4068691)
Affinity DataKi:  0.564nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254132(CHEMBL4083940)
Affinity DataKi:  0.578nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254130(CHEMBL4061334)
Affinity DataKi:  0.585nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254123(CHEMBL4068691)
Affinity DataKi:  0.726nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254122(CHEMBL4098662)
Affinity DataKi:  0.781nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254131(CHEMBL4094845)
Affinity DataKi:  0.813nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254120(CHEMBL4076681)
Affinity DataKi:  0.826nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254120(CHEMBL4076681)
Affinity DataKi:  0.833nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254121(CHEMBL4067629)
Affinity DataKi:  0.953nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254120(CHEMBL4076681)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human recombinant DOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254121(CHEMBL4067629)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254124(CHEMBL4103044)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254122(CHEMBL4098662)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254133(CHEMBL4076632)
Affinity DataEC50:  1.5nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254122(CHEMBL4098662)
Affinity DataEC50:  1.70nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254121(CHEMBL4067629)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254122(CHEMBL4098662)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254120(CHEMBL4076681)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254130(CHEMBL4061334)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254130(CHEMBL4061334)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254130(CHEMBL4061334)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254121(CHEMBL4067629)
Affinity DataEC50:  4.70nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254122(CHEMBL4098662)
Affinity DataEC50:  5.70nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254121(CHEMBL4067629)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254121(CHEMBL4067629)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant MOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254122(CHEMBL4098662)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human recombinant MOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254124(CHEMBL4103044)
Affinity DataEC50:  155nMAssay Description:Agonist activity at human recombinant MOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2019
Entry Details Article
PubMed