Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50049283
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238182BDBM50238182(CHEMBL4100860)
Affinity DataKi:  0.0700nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238177BDBM50238177(CHEMBL4098072)
Affinity DataKi:  0.350nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238162BDBM50238162(CHEMBL4100377)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238182BDBM50238182(CHEMBL4100860)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238157BDBM50238157(CHEMBL4100777)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50322823BDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238193BDBM50238193(CHEMBL4096980)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238172BDBM50238172(CHEMBL4079393)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238165BDBM50238165(CHEMBL4060003)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238177BDBM50238177(CHEMBL4098072)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238181BDBM50238181(CHEMBL4071368)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238160BDBM50238160(CHEMBL4087268)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238173BDBM50238173(CHEMBL4078963)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238185BDBM50238185(CHEMBL4094927)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5447BDBM5447(ZD1839 | N-(3-chloro-4-fluorophenyl)-7-methoxy-6-[...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238186BDBM50238186(CHEMBL4082362)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238191BDBM50238191(CHEMBL4090686)
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238183BDBM50238183(CHEMBL4071012)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029668BDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238183BDBM50238183(CHEMBL4071012)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238174BDBM50238174(CHEMBL4098412)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238159BDBM50238159(CHEMBL4105526)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238192BDBM50238192(CHEMBL4071180)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238168BDBM50238168(CHEMBL4081860)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238170BDBM50238170(CHEMBL4064942)
Affinity DataIC50: 9nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238176BDBM50238176(CHEMBL4091569)
Affinity DataIC50: 11nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383274BDBM50383274(CHEMBL1229592 | US9670213, WZ4002 | US10167264, WZ...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238169BDBM50238169(CHEMBL4062543)
Affinity DataIC50: 12nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029668BDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)
Affinity DataKi:  14nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238161BDBM50238161(CHEMBL4089601)
Affinity DataIC50: 16nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238156BDBM50238156(CHEMBL4089279)
Affinity DataIC50: 16nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238179BDBM50238179(CHEMBL4076854)
Affinity DataIC50: 17nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238164BDBM50238164(CHEMBL4070707)
Affinity DataIC50: 19nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238158BDBM50238158(CHEMBL4102577)
Affinity DataIC50: 22nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238154BDBM50238154(CHEMBL321494)
Affinity DataIC50: 24nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238163BDBM50238163(CHEMBL4061473)
Affinity DataIC50: 28nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238171BDBM50238171(CHEMBL4086878)
Affinity DataIC50: 32nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238184BDBM50238184(CHEMBL4102224)
Affinity DataIC50: 33nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238187BDBM50238187(CHEMBL4084248)
Affinity DataIC50: 45nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238175BDBM50238175(CHEMBL4076363)
Affinity DataIC50: 55nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238188BDBM50238188(CHEMBL4082884)
Affinity DataIC50: 57nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238190BDBM50238190(CHEMBL4081732)
Affinity DataIC50: 109nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238178BDBM50238178(CHEMBL4068092)
Affinity DataIC50: 164nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238155BDBM50238155(CHEMBL4067255)
Affinity DataIC50: 183nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238166BDBM50238166(CHEMBL4092003)
Affinity DataIC50: 185nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238189BDBM50238189(CHEMBL4086078)
Affinity DataIC50: 217nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238167BDBM50238167(CHEMBL4062722)
Affinity DataIC50: 265nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238180BDBM50238180(CHEMBL4101193)
Affinity DataIC50: 1.77E+3nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2019
Entry Details Article
PubMed