Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50000248
TargetAP2-associated protein kinase 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM311218(US10155760, Example 74 | (S)-1-(2-cyclopropyl-4-(q...)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of GST-Xa-tagged human AAK1 expressed in bacterial system using fluoresceinated peptide (5 -FAM)-Aha-KEEQSQITSQVTGQIGWR-NH2 and ATP incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetAP2-associated protein kinase 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM311347(US10155760, Example 204 | (S)-1-((3-(difluoromethy...)
Affinity DataIC50: 0.230nMAssay Description:Inhibition of GST-Xa-tagged human AAK1 expressed in bacterial system using fluoresceinated peptide (5 -FAM)-Aha-KEEQSQITSQVTGQIGWR-NH2 and ATP incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetAP2-associated protein kinase 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM311189(US10155760, Example 33 | (S)-methyl (4-(4-((2-amin...)
Affinity DataIC50: 0.320nMAssay Description:Inhibition of GST-Xa-tagged human AAK1 expressed in bacterial system using fluoresceinated peptide (5 -FAM)-Aha-KEEQSQITSQVTGQIGWR-NH2 and ATP incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetAP2-associated protein kinase 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM311159(BDBM50243381 | US10723734, Example 7 | US9902722, ...)
Affinity DataIC50: 0.420nMAssay Description:Inhibition of GST-Xa-tagged human AAK1 expressed in bacterial system using fluoresceinated peptide (5 -FAM)-Aha-KEEQSQITSQVTGQIGWR-NH2 and ATP incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetAP2-associated protein kinase 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM311266(US10155760, Example 122 | (S)-1-((4-(difluoromethy...)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of GST-Xa-tagged human AAK1 expressed in bacterial system using fluoresceinated peptide (5 -FAM)-Aha-KEEQSQITSQVTGQIGWR-NH2 and ATP incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetAP2-associated protein kinase 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM311154(US10155760, Example 2 | (S)-N-(4-(4-((2-amino-4-me...)
Affinity DataIC50: 3nMAssay Description:Inhibition of GST-Xa-tagged human AAK1 expressed in bacterial system using fluoresceinated peptide (5 -FAM)-Aha-KEEQSQITSQVTGQIGWR-NH2 and ATP incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetAP2-associated protein kinase 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50243380(CHEMBL4066208 | US10544120, Example 337)
Affinity DataIC50: 886nMAssay Description:Inhibition of GST-Xa-tagged human AAK1 expressed in bacterial system using fluoresceinated peptide (5 -FAM)-Aha-KEEQSQITSQVTGQIGWR-NH2 and ATP incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetAP2-associated protein kinase 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM311258(US10155760, Example 114 | (S)-2,4-dimethyl-1-(4-(2...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of GST-Xa-tagged human AAK1 expressed in bacterial system using fluoresceinated peptide (5 -FAM)-Aha-KEEQSQITSQVTGQIGWR-NH2 and ATP incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed