Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50001081
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269051BDBM50269051(CHEMBL4075182)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269062BDBM50269062(CHEMBL4091227)
Affinity DataKi:  4.20nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269087BDBM50269087(CHEMBL4080935)
Affinity DataKi:  4.60nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269075BDBM50269075(CHEMBL4089776)
Affinity DataKi:  7nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269064BDBM50269064(CHEMBL4069278)
Affinity DataKi:  9nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269076BDBM50269076(CHEMBL4077560)
Affinity DataKi:  12nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269043BDBM50269043(CHEMBL4085997)
Affinity DataKi:  18nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269069BDBM50269069(CHEMBL4066184)
Affinity DataKi:  20nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269086BDBM50269086(CHEMBL4075187)
Affinity DataKi:  22nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50050126BDBM50050126((S)-2-((S)-2-Mercapto-3-phenyl-propionylamino)-3-p...)
Affinity DataKi:  23nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269033BDBM50269033(CHEMBL4073385)
Affinity DataKi:  26nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269065BDBM50269065(CHEMBL4066384)
Affinity DataKi:  29nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269035BDBM50269035(CHEMBL4074531)
Affinity DataKi:  30nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269088BDBM50269088(CHEMBL4096514)
Affinity DataKi:  32nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269032BDBM50269032(CHEMBL4094037)
Affinity DataKi:  36nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269063BDBM50269063(CHEMBL4070297)
Affinity DataKi:  36nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269073BDBM50269073(CHEMBL4074608)
Affinity DataKi:  40nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269044BDBM50269044(CHEMBL4087357)
Affinity DataKi:  46nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269050BDBM50269050(CHEMBL4067507)
Affinity DataKi:  49nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269091BDBM50269091(CHEMBL4086067)
Affinity DataKi:  50nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269066BDBM50269066(CHEMBL4088816)
Affinity DataKi:  52nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269049BDBM50269049(CHEMBL4102672)
Affinity DataKi:  54nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269047BDBM50269047(CHEMBL4078411)
Affinity DataKi:  54nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269048BDBM50269048(CHEMBL4095593)
Affinity DataKi:  61nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269060BDBM50269060(CHEMBL4098968)
Affinity DataKi:  61nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269045BDBM50269045(CHEMBL4064153)
Affinity DataKi:  78nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269089BDBM50269089(CHEMBL4088709)
Affinity DataKi:  86nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269031BDBM50269031(CHEMBL4094929)
Affinity DataKi:  95nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269046BDBM50269046(CHEMBL4075680)
Affinity DataKi:  95nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269072BDBM50269072(CHEMBL4100250)
Affinity DataKi:  140nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269074BDBM50269074(CHEMBL4061434)
Affinity DataKi:  162nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269090BDBM50269090(CHEMBL4082357)
Affinity DataKi:  252nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269070BDBM50269070(CHEMBL4101421)
Affinity DataKi:  260nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269067BDBM50269067(CHEMBL4067370)
Affinity DataKi:  470nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269068BDBM50269068(CHEMBL4091335)
Affinity DataKi:  1.65E+3nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269071BDBM50269071(CHEMBL4063351)
Affinity DataKi:  1.75E+3nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetNeprilysin(Human)
Pharmaleads

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269034BDBM50269034(CHEMBL4076819)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human neprilysin using Suc-Ala-Ala-Phe-AMC as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed