Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50049316
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238917(CHEMBL4102009)
Affinity DataIC50:  500nMAssay Description:Opioid receptor mu 1 affinity against the receptor site model site 1 (mu1) by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238926(CHEMBL4081943)
Affinity DataIC50:  640nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238919(CHEMBL4064459)
Affinity DataIC50:  700nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238921(CHEMBL4101461)
Affinity DataIC50:  790nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238913(CHEMBL4076098)
Affinity DataIC50:  830nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238922(CHEMBL4083469)
Affinity DataIC50:  880nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238911(CHEMBL4068882)
Affinity DataIC50:  890nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238918(CHEMBL4102373)
Affinity DataIC50:  940nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238920(CHEMBL4093740)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238915(CHEMBL4064101)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238927(CHEMBL4068968)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238925(CHEMBL4073041)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238916(CHEMBL4083232)
Affinity DataIC50:  2.08E+3nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238924(CHEMBL4078102)
Affinity DataIC50:  2.57E+3nMAssay Description:Opioid receptor mu 2 affinity against the receptor site model site 2(mu2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238914(CHEMBL4073798)
Affinity DataIC50:  3.02E+3nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50238923(CHEMBL4063399)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of human N-terminal His6-tagged QC expressed in Escherichia coli BL21(DE3) using H-gln-gln-H as substrate in presence of NADH/H+ after 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed