Compile Data Set for Download or QSAR
Report error Found 175 Enz. Inhib. hit(s) with all data for entry = 50000834
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261540(CHEMBL4063145)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261540(CHEMBL4063145)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261536(CHEMBL4103639)
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261540(CHEMBL4063145)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261540(CHEMBL4063145)
Affinity DataKi:  0.670nMAssay Description:Agonist activity at human D2SR expressed in HEK293 cell membranes co-expressing PTX insensitive variant of Galphao1 incubated for 30 mins by [35S]GTP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261537(CHEMBL4079375)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261540(CHEMBL4063145)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261540(CHEMBL4063145)
Affinity DataKi:  0.980nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261536(CHEMBL4103639)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261537(CHEMBL4079375)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261537(CHEMBL4079375)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataKi:  1.30nMAssay Description:Agonist activity at human D2SR expressed in HEK293 cell membranes co-expressing PTX insensitive variant of Galphao1 incubated for 30 mins by [35S]GTP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261540(CHEMBL4063145)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261540(CHEMBL4063145)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261536(CHEMBL4103639)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261538(CHEMBL4095881)
Affinity DataKi:  2.90nMAssay Description:Agonist activity at human D2SR expressed in HEK293 cell membranes co-expressing PTX insensitive variant of Galphao1 incubated for 30 mins by [35S]GTP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2AR expressed in HEK293T cell membranes1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261534(CHEMBL4065797)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261538(CHEMBL4095881)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261548(CHEMBL4087217)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261537(CHEMBL4079375)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261542(CHEMBL4085752)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261542(CHEMBL4085752)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261538(CHEMBL4095881)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261542(CHEMBL4085752)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261542(CHEMBL4085752)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261542(CHEMBL4085752)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261542(CHEMBL4085752)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261548(CHEMBL4087217)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261536(CHEMBL4103639)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261531(CHEMBL4084712)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261550(CHEMBL4102646)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261536(CHEMBL4103639)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human D2SR expressed in HEK293 cells incubated for 5 hrs by beta-Arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human D2SR expressed in HEK293 cell membranes co-expressing PTX insensitive variant of Galphao1 incubated for 30 mins by [35S]GTP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261534(CHEMBL4065797)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataEC50:  58nMAssay Description:Agonist activity at human D2SR expressed in HEK293 cell membranes co-expressing PTX insensitive variant of Galphao1 incubated for 30 mins by [35S]GTP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261550(CHEMBL4102646)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261537(CHEMBL4079375)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human D2SR expressed in HEK293 cells incubated for 5 hrs by beta-Arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Friedrich-Alexander University Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50261539(CHEMBL4068561)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human D2SR expressed in HEK293 cells incubated for 5 hrs by beta-Arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/20/2020
Entry Details Article
PubMed
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