Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50001536
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284238(CHEMBL4173941)
Affinity DataIC50:  700nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284239(CHEMBL4161859)
Affinity DataIC50:  800nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284253(CHEMBL4170504)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284252(CHEMBL4166016)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284256(CHEMBL4176982)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284261(CHEMBL4162572)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284251(CHEMBL4174326)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284257(CHEMBL4173619)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM8610(1-[4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imi...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284248(CHEMBL4171198)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284244(CHEMBL4174637)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284199(CHEMBL4159550)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284254(CHEMBL4172837)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284081(CHEMBL4163649)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284249(CHEMBL4160591)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284200(CHEMBL4165064)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284080(CHEMBL4163983)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284264(CHEMBL4159184)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284240(CHEMBL4170175)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284260(CHEMBL4159524)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284263(CHEMBL4162163)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284255(CHEMBL4169784)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284250(CHEMBL4167098)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284143(CHEMBL4166364)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284265(CHEMBL4159101)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284245(CHEMBL4167430)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284237(CHEMBL4169756)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284258(CHEMBL4166769)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284262(CHEMBL4162907)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284241(CHEMBL4168266)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284236(CHEMBL4167841)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284243(CHEMBL4172955)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284191(CHEMBL4170393)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284259(CHEMBL4174670)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Srinakharinwirot University

Curated by ChEMBL
LigandPNGBDBM50284246(CHEMBL4175698)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of aromatase (unknown origin) using O-benzyl fluorescein benzyl ester as substrate in presence of NADPH-generating system by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed