Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50000280
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50244994(CHEMBL4092239)
Affinity DataIC50:  3.20E+3nMAssay Description:Antagonist activity at CXCR4 in human CCRF-CEM cells assessed as inhibition of PE-conjugated 12G5 antibody bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50244999(CHEMBL4094209)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at CXCR4 in human CCRF-CEM cells assessed as inhibition of PE-conjugated 12G5 antibody bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50244997(CHEMBL4070596)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50244998(CHEMBL4064541)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at CXCR4 in human CCRF-CEM cells assessed as inhibition of PE-conjugated 12G5 antibody bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50244995(CHEMBL4083765)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at CXCR4 in human CCRF-CEM cells assessed as inhibition of PE-conjugated 12G5 antibody bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50244996(CHEMBL4101762)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at CXCR4 in human CCRF-CEM cells assessed as inhibition of PE-conjugated 12G5 antibody bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed