Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50006770
Target5-hydroxytryptamine receptor 2C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50161646((R)-8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-benzo[...)
Affinity DataKi:  15nMAssay Description:Agonist activity at 5-HT2CR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 2A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50161646((R)-8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-benzo[...)
Affinity DataKi:  112nMAssay Description:Agonist activity at 5-HT2AR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50161646((R)-8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-benzo[...)
Affinity DataKi:  174nMAssay Description:Agonist activity at 5-HT2BR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
LigandPNGBDBM50503222(CHEMBL4454100)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [3H]-WIN35428 from recombinant human DAT expressed in HEK cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50503222(CHEMBL4454100)
Affinity DataKi:  4.70E+3nMAssay Description:Displacement of [3H]-N-methylspiperone from recombinant human D3R expressed in HEK cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed