Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50002245
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455887(CHEMBL4204982)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to biotinylated HDAC6 ZnF-UBD (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455887(CHEMBL4204982)
Affinity DataIC50: 2.30E+3nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455887(CHEMBL4204982)
Affinity DataIC50: 3.50E+3nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged full length HDAC6 (unknown origin) expressed in Sf9 insec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455900(CHEMBL4215676)
Affinity DataIC50: 5.10E+3nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455900(CHEMBL4215676)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to biotinylated HDAC6 ZnF-UBD (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455896(CHEMBL4206721)
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455892(CHEMBL4218728)
Affinity DataIC50: 4.40E+4nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455886(CHEMBL1416133)
Affinity DataIC50: 4.50E+4nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455902(CHEMBL1708622)
Affinity DataIC50: 5.10E+4nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50242196(CHEMBL4069423)
Affinity DataIC50: 5.50E+4nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50242202(CHEMBL4068652)
Affinity DataIC50: 6.50E+4nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455890(CHEMBL4215552)
Affinity DataIC50: 7.70E+4nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455897(CHEMBL4209794)
Affinity DataIC50: 9.50E+4nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455898(CHEMBL4204813)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455903(CHEMBL1527237)
Affinity DataIC50: 1.50E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455888(CHEMBL4203995)
Affinity DataIC50: 1.80E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455891(CHEMBL4211769)
Affinity DataIC50: 1.90E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455889(CHEMBL4207434)
Affinity DataIC50: 2.00E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455901(CHEMBL284979)
Affinity DataIC50: 2.00E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50234922(CHEMBL1892587)
Affinity DataIC50: 2.30E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455893(CHEMBL4211548)
Affinity DataIC50: 2.40E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455885(CHEMBL1471153)
Affinity DataIC50: 3.20E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455894(CHEMBL4212057)
Affinity DataIC50: 3.90E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455895(CHEMBL4214608)
Affinity DataIC50: 6.40E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50455899(CHEMBL4218506)
Affinity DataIC50: 7.20E+5nMAssay Description:Displacement of N-terminal FITC-labeled RLRGG from N-terminal AviTag/C-terminal His6-tagged HDAC6 ZnF-UBD (unknown origin) expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)