Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50001223
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM220447(US10633379, Compound X | US9296741, 36)
Affinity DataIC50:  1nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50273481(CHEMBL4125931)
Affinity DataIC50:  18nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50273482(CHEMBL4127310)
Affinity DataIC50:  100nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50399434(CHEMBL2179387)
Affinity DataIC50:  220nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataIC50:  630nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50273496(CHEMBL4125924)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50032921(CHEMBL1444120)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50273497(CHEMBL4129632)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50273483(CHEMBL4129169)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50032911(CHEMBL1535485)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50273480(CHEMBL4126342)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50271103(CHEMBL4129770)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50273493(CHEMBL4127163)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50273495(CHEMBL4127306)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50270480(CHEMBL4126540)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50273479(CHEMBL4128551)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bienta/Enamine

Curated by ChEMBL
LigandPNGBDBM50273484(CHEMBL4127934)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed