Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50001483
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50281174(CHEMBL4168736)
Affinity DataKd:  660nMAssay Description:Binding affinity to human HSC70 after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50281174(CHEMBL4168736)
Affinity DataKd:  2.38E+3nMAssay Description:Binding affinity to human HSC70 Y149A mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50281174(CHEMBL4168736)
Affinity DataKd:  5.54E+3nMAssay Description:Binding affinity to human HSC70 Y149W mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50281174(CHEMBL4168736)
Affinity DataKd:  8.25E+3nMAssay Description:Binding affinity to human HSC70 T222A mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50281175(CHEMBL4165078)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human HSC70 after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50281174(CHEMBL4168736)
Affinity DataKd:  1.38E+4nMAssay Description:Binding affinity to human HSC70 L228A mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50281174(CHEMBL4168736)
Affinity DataKd:  2.43E+4nMAssay Description:Binding affinity to human HSC70 H227A mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed