Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50003273
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50: 155nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468904(CHEMBL4173778)
Affinity DataIC50: 309nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468904(CHEMBL4173778)
Affinity DataIC50: 310nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468898(CHEMBL4278309)
Affinity DataIC50: 880nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468898(CHEMBL4278309)
Affinity DataIC50: 891nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468900(CHEMBL4282827)
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468900(CHEMBL4282827)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468901(CHEMBL4294526)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468901(CHEMBL4294526)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468899(CHEMBL4286619)
Affinity DataIC50: 3.69E+3nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468899(CHEMBL4286619)
Affinity DataIC50: 3.72E+3nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468905(CHEMBL4290052)
Affinity DataIC50: 3.66E+4nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein G(o) subunit alpha(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468897(CHEMBL4286220)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant rat Gi coupled mGlu2 receptor expressed in CHO cells assessed as suppression of L-glutamate-induced decrease in cAMP level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein G(o) subunit alpha(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468898(CHEMBL4278309)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant rat Gi coupled mGlu2 receptor expressed in CHO cells assessed as suppression of L-glutamate-induced decrease in cAMP level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein G(o) subunit alpha(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468904(CHEMBL4173778)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant rat Gi coupled mGlu2 receptor expressed in CHO cells assessed as suppression of L-glutamate-induced decrease in cAMP level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468903(CHEMBL4279374)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein G(o) subunit alpha(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468900(CHEMBL4282827)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant rat Gi coupled mGlu2 receptor expressed in CHO cells assessed as suppression of L-glutamate-induced decrease in cAMP level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein subunit alpha-11(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468897(CHEMBL4286220)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human Gq/11 coupled N-terminal 3His-tagged M1 receptor expressed in CHOK1 cells assessed as reduction in carbachol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50468899(CHEMBL4286619)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Gs coupled adrenergic beta2 receptor in HEK293 cells assessed as reduction in isoproterenol-induced cAMP production pretreated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50468903(CHEMBL4279374)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Gs coupled adrenergic beta2 receptor in HEK293 cells assessed as reduction in isoproterenol-induced cAMP production pretreated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50468901(CHEMBL4294526)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Gs coupled adrenergic beta2 receptor in HEK293 cells assessed as reduction in isoproterenol-induced cAMP production pretreated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50468897(CHEMBL4286220)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Gs coupled adrenergic beta2 receptor in HEK293 cells assessed as reduction in isoproterenol-induced cAMP production pretreated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50468904(CHEMBL4173778)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Gs coupled adrenergic beta2 receptor in HEK293 cells assessed as reduction in isoproterenol-induced cAMP production pretreated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50468898(CHEMBL4278309)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Gs coupled adrenergic beta2 receptor in HEK293 cells assessed as reduction in isoproterenol-induced cAMP production pretreated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Gs coupled adrenergic beta2 receptor in HEK293 cells assessed as reduction in isoproterenol-induced cAMP production pretreated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein G(o) subunit alpha(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468903(CHEMBL4279374)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant rat Gi coupled mGlu2 receptor expressed in CHO cells assessed as suppression of L-glutamate-induced decrease in cAMP level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein G(o) subunit alpha(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant rat Gi coupled mGlu2 receptor expressed in CHO cells assessed as suppression of L-glutamate-induced decrease in cAMP level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein G(o) subunit alpha(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468901(CHEMBL4294526)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant rat Gi coupled mGlu2 receptor expressed in CHO cells assessed as suppression of L-glutamate-induced decrease in cAMP level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50468900(CHEMBL4282827)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Gs coupled adrenergic beta2 receptor in HEK293 cells assessed as reduction in isoproterenol-induced cAMP production pretreated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein G(o) subunit alpha(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50468899(CHEMBL4286619)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant rat Gi coupled mGlu2 receptor expressed in CHO cells assessed as suppression of L-glutamate-induced decrease in cAMP level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed