Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50002806
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463302(CHEMBL4239814)
Affinity DataIC50: 0.200nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50431893(ARRY-520 | CHEMBL2347655)
Affinity DataIC50: 6nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463316(KF 89617 | KF-89617 | Kf89617 | LY 2523355 | LY-25...)
Affinity DataIC50: 7nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50431886(CHEMBL1413473)
Affinity DataIC50: 800nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50431886(CHEMBL1413473)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM24174(3-N,3-N-diethyl-5,5-dimethyl-2-N-(thiophene-2-)-4,...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM88776({4-[(5-(4-chlorophenyl)-6-(isopropoxycarbonyl)-7-m...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463314(CHEMBL4246367)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463319(CHEMBL4238439)
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463309(CHEMBL4240281)
Affinity DataIC50: 2.02E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463308(CHEMBL4241043)
Affinity DataIC50: 2.75E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463311(CHEMBL4248454)
Affinity DataIC50: 3.92E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463320(CHEMBL4243218)
Affinity DataIC50: 4.27E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463315(CHEMBL4251458)
Affinity DataIC50: 4.78E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463304(CHEMBL4243138)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463298(CHEMBL4242214)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463301(CHEMBL4247682)
Affinity DataIC50: 6.21E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463310(CHEMBL4246224)
Affinity DataIC50: 6.33E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463305(CHEMBL4247167)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463312(CHEMBL4249742)
Affinity DataIC50: 7.19E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463299(CHEMBL4243604)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463303(CHEMBL4239372)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463318(CHEMBL4246993)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463313(CHEMBL4241249)
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463300(CHEMBL4251217)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463306(CHEMBL4239414)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463307(CHEMBL4244405)
Affinity DataIC50: 1.29E+5nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
University of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463317(CHEMBL4246927)
Affinity DataIC50: 1.34E+5nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed