Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50002832
TargetToll-like receptor 1(Homo sapiens)
Medical University Innsbruck

Curated by ChEMBL
LigandPNGBDBM50463543(CHEMBL4249593)
Affinity DataIC50:  4.58E+4nMAssay Description:Antagonist activity at FLAG-tagged human TLR2/TLR1 expressed in HEK293 cells co-expressing pGL3-Elam.luc assessed as inhibition of Pam3CSK4-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 1/2(Homo sapiens (Human))
Medical University Innsbruck

Curated by ChEMBL
LigandPNGBDBM50463542(CHEMBL4243009)
Affinity DataIC50:  4.92E+4nMAssay Description:Antagonist activity at FLAG-tagged human TLR2/TLR1 expressed in HEK293 cells co-expressing pGL3-Elam.luc assessed as inhibition of Pam3CSK4-stimulate...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed