BindingDB PrimarySearch

Found 72 Enz. Inhib. hit(s) with all data for entry = 50002472

Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458963(CHEMBL4209902)

IC50: 1.10nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458969(CHEMBL4207165)

IC50: 4nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM25121(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,...)

IC50: 4nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458971(CHEMBL4215729)

IC50: 4nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458968(CHEMBL4216442)

IC50: 8.40nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458967(CHEMBL4202820)

IC50: 8.60nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458960(CHEMBL4216875)

IC50: 8.70nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458962(CHEMBL4213276)

IC50: 9nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458951(CHEMBL4206171)

IC50: 9.90nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458965(CHEMBL4210571)

IC50: 21nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458964(CHEMBL4206052)

IC50: 25nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458952(CHEMBL4203571)

IC50: 27nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458966(CHEMBL4207437)

IC50: 28nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 32nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50112336(CHEMBL3609305)

IC50: 33nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458959(CHEMBL4214823)

IC50: 37nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458966(CHEMBL4207437)

IC50: 40nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458955(CHEMBL4209192)

IC50: 47nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50112335(CHEMBL3609304)

IC50: 54nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458970(CHEMBL4206381)

IC50: 59nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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B.MOAD antibodypedia GoogleScholar

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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458958(CHEMBL4215910)

IC50: 78nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458963(CHEMBL4209902)

IC50: 84nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458956(CHEMBL4202678)

IC50: 94nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458968(CHEMBL4216442)

IC50: 95nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458956(CHEMBL4202678)

IC50: 95nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Bromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458966(CHEMBL4207437)

IC50: 102nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Bromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 103nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB MMDB KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458965(CHEMBL4210571)

IC50: 104nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458960(CHEMBL4216875)

IC50: 107nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458961(CHEMBL4210414)

IC50: 107nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458962(CHEMBL4213276)

IC50: 109nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458970(CHEMBL4206381)

IC50: 127nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458961(CHEMBL4210414)

IC50: 160nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458952(CHEMBL4203571)

IC50: 183nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458969(CHEMBL4207165)

IC50: 186nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM25121(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,...)

IC50: 205nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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3D Structure (crystal)

Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458957(CHEMBL4212237)

IC50: 218nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Bromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458960(CHEMBL4216875)

IC50: 229nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
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Bromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458970(CHEMBL4206381)

IC50: 245nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458973(CHEMBL4212346)

IC50: 253nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Bromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458968(CHEMBL4216442)

IC50: 289nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458967(CHEMBL4202820)

IC50: 310nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458954(CHEMBL4207347)

IC50: 322nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Bromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458963(CHEMBL4209902)

IC50: 342nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB MMDB KEGG
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Bromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458956(CHEMBL4202678)

IC50: 369nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB MMDB KEGG
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Bromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458961(CHEMBL4210414)

IC50: 378nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB MMDB KEGG
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Bromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458965(CHEMBL4210571)

IC50: 392nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458964(CHEMBL4206052)

IC50: 421nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Serine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50458973(CHEMBL4212346)

IC50: 457nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston

Curated by ChEMBL

BDBM50112336(CHEMBL3609305)

IC50: 489nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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