TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 501nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2 cells incubated for 30 mins measured at 60 secs interval for 120 mins by Hoechst 33342 staini...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 526nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 731nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 940nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in HEK293 cells assessed as reduction in mitoxantrone efflux measured after 30 mins by fluorescence as...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in HEK293 cells assessed as reduction in mitoxantrone efflux measured after 30 mins by fluorescence as...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 2.13E+3nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 2.83E+3nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 4.08E+3nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 6.65E+3nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 6.73E+3nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 8.76E+3nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Universidad Nacional De Colombia-Sede Bogot£
Curated by ChEMBL
Affinity DataIC50: 2.32E+4nMAssay Description:Inhibition of ABCG2 in human MCF7/Topo cells after 2 hrs by Hoechst 33342 staining based fluorescence assayMore data for this Ligand-Target Pair