Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50003104
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467028(CHEMBL4281089)
Affinity DataIC50:  900nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467029(CHEMBL4285364)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467033(CHEMBL4279547)
Affinity DataIC50:  6.90E+3nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467030(CHEMBL4290212)
Affinity DataIC50:  7.60E+3nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50:  2.20E+4nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467032(CHEMBL4284935)
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed