TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases
Curated by ChEMBL
Janssen Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases
Curated by ChEMBL
Janssen Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases
Curated by ChEMBL
Janssen Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases
Curated by ChEMBL
Janssen Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases
Curated by ChEMBL
Janssen Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Infectious Diseases
Curated by ChEMBL
Janssen Infectious Diseases
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair