Compile Data Set for Download or QSAR
maximum 50k data
Found 107 Enz. Inhib. hit(s) with all data for entry = 50002511
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459512(CHEMBL4211240)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human KLK6 expressed in baculovirus/insect cell line system using Abz-KLRSSKQ-EDDnp substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)
Affinity DataIC50: <1nMAssay Description:Inhibition of trypsin (unknown origin) pre-incubated for 30 mins before N-Boc-FSR-AMC substrate addition and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)
Affinity DataIC50:  8nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459537(CHEMBL4217078)
Affinity DataIC50:  18nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)
Affinity DataIC50:  23nMAssay Description:Inhibition of KLK6 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459515(CHEMBL4216138)
Affinity DataIC50:  100nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459525(CHEMBL4212718)
Affinity DataIC50:  100nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459545(CHEMBL4210314)
Affinity DataIC50:  130nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)
Affinity DataIC50:  130nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459538(CHEMBL4218203)
Affinity DataIC50:  130nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459527(CHEMBL4203947)
Affinity DataIC50:  150nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459529(CHEMBL4208878)
Affinity DataIC50:  180nMAssay Description:Inhibition of trypsin (unknown origin) pre-incubated for 30 mins before N-Boc-FSR-AMC substrate addition and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459508(CHEMBL4211164)
Affinity DataIC50:  190nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-8(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)
Affinity DataIC50:  210nMAssay Description:Inhibition of KLK8 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459531(CHEMBL4207925)
Affinity DataIC50:  250nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459535(CHEMBL4214705)
Affinity DataIC50:  250nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459522(CHEMBL4218314)
Affinity DataIC50:  290nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459515(CHEMBL4216138)
Affinity DataIC50:  330nMAssay Description:Inhibition of trypsin (unknown origin) pre-incubated for 30 mins before N-Boc-FSR-AMC substrate addition and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459537(CHEMBL4217078)
Affinity DataIC50:  380nMAssay Description:Inhibition of trypsin (unknown origin) pre-incubated for 30 mins before N-Boc-FSR-AMC substrate addition and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459538(CHEMBL4218203)
Affinity DataIC50:  470nMAssay Description:Inhibition of KLK6 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459516(CHEMBL4211677)
Affinity DataIC50:  490nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)
Affinity DataIC50: >500nMAssay Description:Inhibition of KLK7 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Leu-Leu-Val-Tyr-AMC substrate addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-13(Homo sapiens)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)
Affinity DataIC50: >500nMAssay Description:Inhibition of KLK13 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459511(CHEMBL4212332)
Affinity DataIC50:  640nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459529(CHEMBL4208878)
Affinity DataIC50:  890nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459538(CHEMBL4218203)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459526(CHEMBL4218619)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459541(CHEMBL4204137)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459524(CHEMBL4215806)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459520(CHEMBL4203193)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459526(CHEMBL4218619)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of trypsin (unknown origin) pre-incubated for 30 mins before N-Boc-FSR-AMC substrate addition and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459543(CHEMBL4203033)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459507(CHEMBL4215383)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459546(CHEMBL4206799)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459514(CHEMBL4205963)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459548(CHEMBL4210959)
Affinity DataIC50:  6.99E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459523(CHEMBL4206590)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459542(CHEMBL4212830)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459543(CHEMBL4203033)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of trypsin (unknown origin) pre-incubated for 30 mins before N-Boc-FSR-AMC substrate addition and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459544(CHEMBL4217674)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459536(CHEMBL4211986)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-13(Homo sapiens)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459538(CHEMBL4218203)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of KLK13 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-8(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459538(CHEMBL4218203)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of KLK8 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459509(CHEMBL1883669)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-14(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459538(CHEMBL4218203)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459530(CHEMBL4210322)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459547(CHEMBL4205435)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459534(CHEMBL4206077)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 pre-incubated for 30 mins before N-Boc-FSR-AMC substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459525(CHEMBL4212718)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of trypsin (unknown origin) pre-incubated for 30 mins before N-Boc-FSR-AMC substrate addition and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459538(CHEMBL4218203)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of trypsin (unknown origin) pre-incubated for 30 mins before N-Boc-FSR-AMC substrate addition and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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