BindingDB PrimarySearch_ki

Found 136 Enz. Inhib. hit(s) with all data for entry = 50002517

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)

Ki: 5.30nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed DrugBank
PDB

3D Structure (crystal)

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459619(CHEMBL4206824)

Ki: 6.70nMAssay Description:Displacement of [125I]DOI from human 5HT2A receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase PC cid PC sid

Details Article PubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)

Ki: 11nMAssay Description:Displacement of [125I]DOI from human 5HT2A receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)

Ki: 12nMAssay Description:Displacement of [125I]DOI from human 5HT2A receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL KEGG PC cid PC sid PDB Similars

Details Article PubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459626(CHEMBL4214975)

Ki: 37nMAssay Description:Displacement of [125I]DOI from human 5HT2A receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459625(CHEMBL4205254)

Ki: 62nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459625(CHEMBL4205254)

Ki: 62nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50192902(2-ethyl-3-isobutyl-9,10-dimethoxy-2,3,4,6,7,11b-he...)

Ki: 64nMAssay Description:Displacement of [3H]DHTB from human VMAT2 expressed in HEK293 cell membranes incubated for 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459619(CHEMBL4206824)

Ki: 70nMAssay Description:Displacement of [3H]DHTB from human VMAT2 expressed in HEK293 cell membranes incubated for 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase PC cid PC sid

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459630(CHEMBL4207658)

Ki: 70nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459621(CHEMBL4202787)

Ki: 74nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)

Ki: 77nMAssay Description:Displacement of [3H]DHTB from human VMAT2 expressed in HEK293 cell membranes incubated for 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed PDB

3D Structure (crystal)

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50192902(2-ethyl-3-isobutyl-9,10-dimethoxy-2,3,4,6,7,11b-he...)

Ki: 83nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459619(CHEMBL4206824)

Ki: 152nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase PC cid PC sid

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459621(CHEMBL4202787)

Ki: 161nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459626(CHEMBL4214975)

Ki: 176nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459630(CHEMBL4207658)

Ki: 287nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459625(CHEMBL4205254)

Ki: 290nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459627(CHEMBL4208779)

Ki: 350nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)

Ki: 353nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed PDB

3D Structure (crystal)

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)

Ki: 410nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed DrugBank
PDB

3D Structure (crystal)

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459628(CHEMBL4208250)

Ki: 450nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459618(CHEMBL4216117)

Ki: 452nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)

Ki: 630nMAssay Description:Displacement of [3H]DHTB from human VMAT2 expressed in HEK293 cell membranes incubated for 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed DrugBank
PDB

3D Structure (crystal)

Sodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)

Ki: 632nMAssay Description:Displacement of [125I]RTI-55 from human SERT expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
DrugBank KEGG MMDB PC cid PC sid PDB Patents Similars

Details Article PubMed DrugBank
PDB

3D Structure (crystal)

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459617(CHEMBL4213176)

Ki: 652nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459617(CHEMBL4213176)

Ki: 700nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459624(CHEMBL4203894)

Ki: 720nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459626(CHEMBL4214975)

Ki: 750nMAssay Description:Displacement of [3H]DHTB from human VMAT2 expressed in HEK293 cell membranes incubated for 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459628(CHEMBL4208250)

Ki: 900nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459627(CHEMBL4208779)

Ki: 990nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)

Ki: >1.00E+3nMAssay Description:Displacement of [125I]DOI from human 5HT2A receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459626(CHEMBL4214975)

Ki: 1.15E+3nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)

Ki: 1.19E+3nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed PDB

3D Structure (crystal)

Sodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459630(CHEMBL4207658)

Ki: 1.61E+3nMAssay Description:Displacement of [125I]RTI-55 from human DAT expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459622(CHEMBL4217581)

Ki: 1.66E+3nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50080818((-)-lobeline | 2-(6-(2-Hydroxy-2-phenylethyl)-1-me...)

Ki: 1.84E+3nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG MMDB PC cid PC sid PDB Patents Similars

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50192902(2-ethyl-3-isobutyl-9,10-dimethoxy-2,3,4,6,7,11b-he...)

Ki: 1.93E+3nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50080818((-)-lobeline | 2-(6-(2-Hydroxy-2-phenylethyl)-1-me...)

Ki: 1.95E+3nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG MMDB PC cid PC sid PDB Patents Similars

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459620(CHEMBL4204449)

Ki: 1.96E+3nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)

Ki: 2.29E+3nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL KEGG PC cid PC sid PDB Similars

Details Article PubMed PDB

3D Structure (crystal)

Sodium-dependent noradrenaline transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)

Ki: 2.36E+3nMAssay Description:Displacement of [125I]RTI-55 from human NET expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase ChEBI
DrugBank KEGG MMDB PC cid PC sid PDB Patents Similars

Details Article PubMed DrugBank

5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459621(CHEMBL4202787)

Ki: 2.38E+3nMAssay Description:Displacement of [125I]DOI from human 5HT2A receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Sodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459625(CHEMBL4205254)

Ki: 2.44E+3nMAssay Description:Displacement of [125I]RTI-55 from human DAT expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar

Details Article PubMed

Sodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459625(CHEMBL4205254)

Ki: 2.44E+3nMAssay Description:Displacement of [125I]RTI-55 from human DAT expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459623(CHEMBL4212633)

Ki: 3.77E+3nMAssay Description:Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 e...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Sodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459621(CHEMBL4202787)

Ki: 4.17E+3nMAssay Description:Displacement of [125I]RTI-55 from human DAT expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459628(CHEMBL4208250)

Ki: 6.16E+3nMAssay Description:Displacement of [3H]DHTB from human VMAT2 expressed in HEK293 cell membranes incubated for 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Synaptic vesicular amine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50009057((R)Methyl-(1-methyl-2-phenyl-ethyl)-amine | METHAM...)

Ki: 6.40E+3nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase PC cid PC sid PDB Patents Similars

Details Article PubMed

Sodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL

PNG

BDBM50459628(CHEMBL4208250)

Ki: >7.10E+3nMAssay Description:Displacement of [125I]RTI-55 from human DAT expressed in HEK293 cell membranesMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar

Details Article PubMed

Displayed 1 to 50 (of 136 total ) | Next | Last >>