Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for entry = 50002527
TargetHistone deacetylase 1(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50459720(CHEMBL4210305)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of recombinant human C-terminal FLAG/His-tagged HDAC1 expressed in baculovirus infected Sf9 insect cells using HDAC substrate 3 measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50459720(CHEMBL4210305)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of recombinant human C-terminal FLAG-tagged HDAC2 expressed in baculovirus infected Sf9 insect cells using HDAC substrate 3 measured after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50459720(CHEMBL4210305)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human full length C-terminal His-tagged HDAC3/N-terminal GST-tagged human NCOR2 (395 to 489 residues) co-expressed in baculovirus infec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Kansai University

Curated by ChEMBL
LigandPNGBDBM50459720(CHEMBL4210305)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of human HDAC10 expressed in baculovirus infected Sf9 insect cells using HDAC substrate 3 measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed