TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Anhui University Of Chinese Medicine
Curated by ChEMBL
Anhui University Of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of MDR1 in human KB/VCR cells assessed as potentiation of vincristine-induced cytotoxicity by measuring vincristine IC50 at 25 uM after 72...More data for this Ligand-Target Pair