Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50048759
LigandChemical structure of BindingDB Monomer ID 50226932BDBM50226932(CHEMBL559829)
Affinity DataKi:  6.60nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226924BDBM50226924(CHEMBL545647)
Affinity DataKi:  6.90nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50019848BDBM50019848(CHEMBL10316 | Idazoxan | US8633208, Idazoxan | 4,5...)
Affinity DataKi:  10nMAssay Description:Ability to displace [3H]-clonidine from alpha-1 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50019848BDBM50019848(CHEMBL10316 | Idazoxan | US8633208, Idazoxan | 4,5...)
Affinity DataKi:  10nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226929BDBM50226929(CHEMBL545646)
Affinity DataKi:  12nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226929BDBM50226929(CHEMBL545646)
Affinity DataKi:  12nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50454831BDBM50454831(Napamezole)
Affinity DataKi:  23nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50454831BDBM50454831(Napamezole)
Affinity DataKi:  23nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226928BDBM50226928(CHEMBL553439)
Affinity DataKi:  32nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50057120BDBM50057120(cid_610682 | CHEMBL441948 | 2-Naphthalen-2-ylmethy...)
Affinity DataKi:  48nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50222218BDBM50222218(CHEBI:51137 | Mianserin)
Affinity DataKi:  76nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226927BDBM50226927(CHEMBL544701)
Affinity DataKi:  76nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50454831BDBM50454831(Napamezole)
Affinity DataKi:  78nMAssay Description:Ability to displace [3H]prazosin from alpha-1 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50013515BDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  78nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226930BDBM50226930(CHEMBL35345)
Affinity DataKi:  88nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226926BDBM50226926(CHEMBL544706)
Affinity DataKi:  135nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226929BDBM50226929(CHEMBL545646)
Affinity DataKi:  148nMAssay Description:Ability to displace [3H]prazosin from alpha-1 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50019848BDBM50019848(CHEMBL10316 | Idazoxan | US8633208, Idazoxan | 4,5...)
Affinity DataKi:  261nMAssay Description:Ability to displace [3H]prazosin from alpha-1 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226921BDBM50226921(CHEMBL544704)
Affinity DataKi:  334nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226923BDBM50226923(CHEMBL544705)
Affinity DataKi:  401nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226925BDBM50226925(CHEMBL553103)
Affinity DataKi:  436nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226931BDBM50226931(CHEMBL553368)
Affinity DataKi:  548nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226922BDBM50226922(CHEMBL543535)
Affinity DataKi: >800nMAssay Description:Ability to displace [3H]clonidine from alpha-2 adrenergic receptor in rat brain homogenates in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed