Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50022565
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50064091((2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataEC50:  25nMAssay Description:Activation of PKC in human ACH-2 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50064091((2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataEC50:  34nMAssay Description:Activation of PKC in human U1 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50057511(CHEMBL27266 | 13-Hydroxymethyl-10-isopropyl-9-meth...)
Affinity DataEC50:  47nMAssay Description:Activation of PKC in human ACH-2 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50368315(PROSTRATIN)
Affinity DataEC50:  280nMAssay Description:Activation of PKC in human U1 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50368315(PROSTRATIN)
Affinity DataEC50:  294nMAssay Description:Activation of PKC in human ACH-2 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50057511(CHEMBL27266 | 13-Hydroxymethyl-10-isopropyl-9-meth...)
Affinity DataEC50:  360nMAssay Description:Activation of PKC in human U1 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50652926(CHEMBL5678793)
Affinity DataEC50:  430nMAssay Description:Activation of PKC in human ACH-2 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50652927(CHEMBL5678789)
Affinity DataEC50:  1.54E+3nMAssay Description:Activation of PKC in human ACH-2 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50652926(CHEMBL5678793)
Affinity DataEC50:  2.33E+3nMAssay Description:Activation of PKC in human U1 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50064095((7S,10S)-10-Hydroxymethyl-7-isopropyl-1,1,4,4,6-pe...)
Affinity DataEC50:  2.91E+3nMAssay Description:Activation of PKC in human ACH-2 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50652927(CHEMBL5678789)
Affinity DataEC50:  4.00E+3nMAssay Description:Activation of PKC in human U1 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50064091((2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataEC50:  6.30E+3nMAssay Description:Activation of PKC in human J-Lat 6.3 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase of GFP-positive cel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50064095((7S,10S)-10-Hydroxymethyl-7-isopropyl-1,1,4,4,6-pe...)
Affinity DataEC50:  9.89E+3nMAssay Description:Activation of PKC in human U1 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase in p24 antigen level incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50064091((2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataEC50:  1.06E+4nMAssay Description:Activation of PKC in human J-Lat 10.6 cells infected with latent HIV-1 assessed as reversal of HIV-1 latency by measuring increase of GFP-positive ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed