TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human N-terminal GST-tagged HDAC7 (518 to end residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substra...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human C-terminal His-tagged HDAC9 (604 to 1066 residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substr...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of human N-terminal GST-tagged HDAC7 (518 to end residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substra...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human C-terminal His-tagged HDAC9 (604 to 1066 residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substr...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human N-terminal GST-tagged HDAC7 (518 to end residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substra...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 103nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 119nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human C-terminal His-tagged HDAC9 (604 to 1066 residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substr...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of HDAC4 catalytic domain (648 to 1057 residues) (unknown origin) using Boc-Lys-TFA as substrate measured after 60 mins by fluorescence as...More data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of human C-terminal His-tagged HDAC9 (604 to 1066 residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substr...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of human N-terminal GST-tagged HDAC7 (518 to end residues) expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substra...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of recombinant human HDAC6 expressed in HEK293 cells using Lys-Ac-AMC as substrate measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of recombinant human HDAC6 expressed in HEK293 cells using Lys-Ac-AMC as substrate measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of recombinant human HDAC6 expressed in HEK293 cells using Lys-Ac-AMC as substrate measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human full length C-terminal His-tagged HDAC8 expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substrate measure...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of human full length C-terminal His-tagged HDAC8 expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substrate measure...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]dofetilide from recombinant human ERG after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human HDAC6 expressed in HEK293 cells using Lys-Ac-AMC as substrate measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of human full length C-terminal His-tagged HDAC8 expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substrate measure...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of HDAC6 in human A549 cells using tubulin as substrate measured after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of full length recombinant human C-terminal His-tagged HDAC3/N-terminal GST-tagged NCOR2 co-expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 2.58E+4nMAssay Description:Inhibition of full length recombinant human C-terminal His-tagged HDAC3/N-terminal GST-tagged NCOR2 co-expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
TargetHistone deacetylase 1/2/3/8(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of HDAC class 1 in human A549 cells using histone H4K12 as substrate measured after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 3.89E+4nMAssay Description:Inhibition of full length recombinant human C-terminal His-tagged HDAC3/N-terminal GST-tagged NCOR2 co-expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 3.97E+4nMAssay Description:Inhibition of human full length C-terminal FLAG/His-tagged HDAC1 expressed in baculovirus infected Sf9 insect cells using Lys-Ac-AMC as substrate mea...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of human full length C-terminal His-tagged HDAC8 expressed in baculovirus infected Sf9 insect cells using Boc-Lys-TFA as substrate measure...More data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of full length recombinant human C-terminal His-tagged HDAC3/N-terminal GST-tagged NCOR2 co-expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human full length C-terminal FLAG-tagged HDAC2 expressed in baculovirus infected Sf9 insect cells using Ac-Arg-Gly-Lys(Ac) as substrate...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Charles River Discovery (Previously Biofocus)
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human full length C-terminal FLAG-tagged HDAC2 expressed in baculovirus infected Sf9 insect cells using Ac-Arg-Gly-Lys(Ac) as substrate...More data for this Ligand-Target Pair