Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50008655
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50521197(CHEMBL4550460)
Affinity DataIC50:  1.85E+4nMAssay Description:Antagonist activity at human TRPM8 channel expressed in HEK293 cells assessed as inhibition of icilin-induced calcium flux by Fluo-4-AM dye based flu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50521199(CHEMBL4513622)
Affinity DataIC50:  4.59E+4nMAssay Description:Antagonist activity at human TRPV4 channel expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced calcium flux by Fluo-4-AM dye base...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50521198(CHEMBL4533807)
Affinity DataIC50:  6.16E+4nMAssay Description:Antagonist activity at human TRPM8 channel expressed in HEK293 cells assessed as inhibition of icilin-induced calcium flux by Fluo-4-AM dye based flu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50521199(CHEMBL4513622)
Affinity DataIC50:  8.16E+4nMAssay Description:Antagonist activity at human TRPV1 channel expressed in human BEAS2B cells assessed as inhibition of capsaicin-induced calcium flux by Fluo-4-AM dye ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed