Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50009179
TargetP2X purinoceptor 7(Homo sapiens (Human))
Fluminense Federal University

Curated by ChEMBL
LigandPNGBDBM50525941(CHEMBL4445773)
Affinity DataIC50:  103nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 5 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Fluminense Federal University

Curated by ChEMBL
LigandPNGBDBM50525940(CHEMBL4454986)
Affinity DataIC50:  230nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 5 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Fluminense Federal University

Curated by ChEMBL
LigandPNGBDBM50234965(A-740003 | CHEMBL255787 | N-(1-(2-cyano-3-(quinoli...)
Affinity DataIC50:  750nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 5 mins fol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Fluminense Federal University

Curated by ChEMBL
LigandPNGBDBM50277548(CHEMBL4173394)
Affinity DataIC50:  1.37E+3nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 5 mins fol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed