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Found 22 Enz. Inhib. hit(s) with all data for entry = 50008386
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518668(CHEMBL4546569)
Affinity DataIC50:  32nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518676(CHEMBL4453888)
Affinity DataIC50:  94nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518675(CHEMBL4458898)
Affinity DataIC50:  280nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518679(CHEMBL4468962)
Affinity DataIC50:  640nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518673(CHEMBL4448964)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518665(CHEMBL4445587)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518667(CHEMBL4585746)
Affinity DataIC50:  1.94E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518661(CHEMBL4554148)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518666(CHEMBL4556590)
Affinity DataIC50:  2.79E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518671(CHEMBL4560122)
Affinity DataIC50:  3.24E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518680(CHEMBL4573946)
Affinity DataIC50:  4.05E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518677(CHEMBL4467680)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518664(CHEMBL4473863)
Affinity DataIC50:  5.41E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518678(CHEMBL4516802)
Affinity DataIC50:  6.38E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM37953(US10093631, Compound Lesinurad | US10336710, Lesin...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM37953(US10093631, Compound Lesinurad | US10336710, Lesin...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of human URAT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518662(CHEMBL4436938)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518663(CHEMBL4551589)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518670(CHEMBL4568207)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518669(CHEMBL4517057)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518672(CHEMBL4594032)
Affinity DataIC50:  1.19E+5nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518674(CHEMBL4459618)
Affinity DataIC50:  3.65E+5nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed