TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of ABCB1 in human A2780/ADR cells preincubated for 30 mins followed by calcein AM addition and measured every 60 secs for 1 hr by fluoresc...More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of ABCB1 in human A2780/ADR cells preincubated for 30 mins followed by calcein AM addition and measured every 60 secs for 1 hr by fluoresc...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 3.37E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 3.58E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 3.75E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 4.28E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 4.74E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 4.91E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of ABCB1 in human A2780/ADR cells preincubated for 30 mins followed by calcein AM addition and measured every 60 secs for 1 hr by fluoresc...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 5.09E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 5.43E+3nMAssay Description:Inhibition of ABCB1 in human A2780/ADR cells preincubated for 30 mins followed by calcein AM addition and measured every 60 secs for 1 hr by fluoresc...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 6.08E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 6.11E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 6.33E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 6.44E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 6.63E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 6.89E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 6.95E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 7.22E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 7.29E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 8.44E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 9.21E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 9.93E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of ABCB1 in human A2780/ADR cells preincubated for 30 mins followed by calcein AM addition and measured every 60 secs for 1 hr by fluoresc...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of ABCC1 in human H96AR cells preincubated for 30 mins followed by calcein AM addition and measured every 60 secs for 1 hr by fluorescence...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.62E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 2.01E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK II BCRP cells assessed as effect on pheophorbide A accumulation after 120 mins by flow cytomet...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataEC50: 1.22E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2 cells co-expressing BCRP (unknown origin) assessed as potentiation of SN-38-induced cytotoxic...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataEC50: 793nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2 cells co-expressing BCRP (unknown origin) assessed as potentiation of SN-38-induced cytotoxic...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataEC50: 1.39E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2 cells co-expressing BCRP (unknown origin) assessed as potentiation of SN-38-induced cytotoxic...More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataEC50: 89nMAssay Description:Inhibition of ABCB1 in human A2780/ADR cells assessed as potentiation of daunorubicin-induced cytotoxicity measured after 72 hrs by MTT assayMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataEC50: 2.09E+3nMAssay Description:Inhibition of ABCB1 in human A2780/ADR cells assessed as potentiation of daunorubicin-induced cytotoxicity measured after 72 hrs by MTT assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataEC50: 1.17E+3nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2 cells co-expressing BCRP (unknown origin) assessed as potentiation of SN-38-induced cytotoxic...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataEC50: 104nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2 cells co-expressing BCRP (unknown origin) assessed as potentiation of SN-38-induced cytotoxic...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataEC50: 446nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2 cells co-expressing BCRP (unknown origin) assessed as potentiation of SN-38-induced cytotoxic...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataEC50: 448nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2 cells co-expressing BCRP (unknown origin) assessed as potentiation of SN-38-induced cytotoxic...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataEC50: 107nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2 cells co-expressing BCRP (unknown origin) assessed as potentiation of SN-38-induced cytotoxic...More data for this Ligand-Target Pair