Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50022625
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Virginia Commonwealth University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50514308(CHEMBL4448899)
Affinity DataIC50: 25nMAssay Description:Inhibition of GLUT1 in human HEY cells assessed as decrease in conversion of D-[5-3H(N)]-glucose to 3H2O incubated for 24 hrs by liquid scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Virginia Commonwealth University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50514308(CHEMBL4448899)
Affinity DataIC50: 25nMAssay Description:Inhibition of GLUT1 in human OVCAR-3 cells assessed as decrease in conversion of D-[5-3H(N)]-glucose to 3H2O incubated for 24 hrs by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Virginia Commonwealth University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50514308(CHEMBL4448899)
Affinity DataIC50: 25nMAssay Description:Inhibition of GLUT1 in human SK-OV-3 cells assessed as decrease in conversion of D-[5-3H(N)]-glucose to 3H2O incubated for 24 hrs by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Virginia Commonwealth University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50514308(CHEMBL4448899)
Affinity DataIC50: 25nMAssay Description:Inhibition of GLUT1 in human OVCA-432 cells assessed as decrease in conversion of D-[5-3H(N)]-glucose to 3H2O incubated for 24 hrs by liquid scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Virginia Commonwealth University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50514308(CHEMBL4448899)
Affinity DataIC50: 25nMAssay Description:Inhibition of GLUT1 in human OVCR-429 cells assessed as decrease in conversion of D-[5-3H(N)]-glucose to 3H2O incubated for 24 hrs by liquid scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed