Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50008400
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518789(CHEMBL4473548)
Affinity DataIC50:  330nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged VEGFR2 (D807 to V1356 residues) expressed in sf9 cells using Poly(Glu,Tyr) 4:1 as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlcohol dehydrogenase 1A(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518790(CHEMBL4465918)
Affinity DataIC50:  460nMAssay Description:Inhibition of ADH1 (unknown origin) preincubated for 2 hrs followed by substrate/NAD+ additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518790(CHEMBL4465918)
Affinity DataIC50:  530nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged VEGFR2 (D807 to V1356 residues) expressed in sf9 cells using Poly(Glu,Tyr) 4:1 as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518789(CHEMBL4473548)
Affinity DataIC50:  540nMAssay Description:Inhibition of recombinant human N-terminal GST/His6-tagged ABL2 (M1 to P650 residues) expressed in sf9 cells using Poly(Glu,Tyr) 4:1 as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518790(CHEMBL4465918)
Affinity DataIC50:  685nMAssay Description:Inhibition of recombinant human N-terminal GST/His6-tagged ABL2 (M1 to P650 residues) expressed in sf9 cells using Poly(Glu,Tyr) 4:1 as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518790(CHEMBL4465918)
Affinity DataIC50:  1.28E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged VEGFR1 (K784 to I1338 residues) expressed in sf9 cells using Poly(Glu,Tyr) 4:1 as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518789(CHEMBL4473548)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged VEGFR1 (K784 to I1338 residues) expressed in sf9 cells using Poly(Glu,Tyr) 4:1 as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518790(CHEMBL4465918)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST/His6-tagged c-KIT (T544 to V976 residues) expressed in sf9 cells using Poly(Glu,Tyr) 4:1 as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518790(CHEMBL4465918)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of recombinant human N-terminal GST/His6-tagged VEGFR3 (N799 to R1298 residues) expressed in sf9 cells using Poly(Glu,Tyr) 4:1 as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlcohol dehydrogenase 1A(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518789(CHEMBL4473548)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of ADH1 (unknown origin) preincubated for 2 hrs followed by substrate/NAD+ additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518789(CHEMBL4473548)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of recombinant human N-terminal GST/His6-tagged c-KIT (T544 to V976 residues) expressed in sf9 cells using Poly(Glu,Tyr) 4:1 as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50518789(CHEMBL4473548)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST/His6-tagged VEGFR3 (N799 to R1298 residues) expressed in sf9 cells using Poly(Glu,Tyr) 4:1 as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed