Compile Data Set for Download or QSAR
Report error Found 502 Enz. Inhib. hit(s) with all data for entry = 50009566
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105834BDBM50105834(CHEMBL3597594)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105834BDBM50105834(CHEMBL3597594)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529980BDBM50529980(CHEMBL4535926)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529958BDBM50529958(CHEMBL4472693)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529980BDBM50529980(CHEMBL4535926)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529958BDBM50529958(CHEMBL4472693)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105834BDBM50105834(CHEMBL3597594)
Affinity DataIC50: 0.800nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in CHO-TREx cell membranes assessed as reduction in quisqualate-induced Ca2+ mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105834BDBM50105834(CHEMBL3597594)
Affinity DataIC50: 0.800nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in CHO-TREx cell membranes assessed as reduction in quisqualate-induced Ca2+ mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529979BDBM50529979(CHEMBL4439229)
Affinity DataKi:  0.980nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529979BDBM50529979(CHEMBL4439229)
Affinity DataKi:  0.980nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529954BDBM50529954(CHEMBL4446275)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529954BDBM50529954(CHEMBL4446275)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529958BDBM50529958(CHEMBL4472693)
Affinity DataIC50: 2.5nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in CHO-TREx cell membranes assessed as reduction in quisqualate-induced Ca2+ mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529958BDBM50529958(CHEMBL4472693)
Affinity DataIC50: 2.5nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in CHO-TREx cell membranes assessed as reduction in quisqualate-induced Ca2+ mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529965BDBM50529965(CHEMBL4441707)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529965BDBM50529965(CHEMBL4441707)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529962BDBM50529962(CHEMBL4539036)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529962BDBM50529962(CHEMBL4539036)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529972BDBM50529972(CHEMBL4472416)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529972BDBM50529972(CHEMBL4472416)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529976BDBM50529976(CHEMBL4452522)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529976BDBM50529976(CHEMBL4452522)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529977BDBM50529977(CHEMBL4451661)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529978BDBM50529978(CHEMBL4592284)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529977BDBM50529977(CHEMBL4451661)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529957BDBM50529957(CHEMBL4455843)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529957BDBM50529957(CHEMBL4455843)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529978BDBM50529978(CHEMBL4592284)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529973BDBM50529973(CHEMBL4513498)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529965BDBM50529965(CHEMBL4441707)
Affinity DataIC50: 3.30nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in CHO-TREx cell membranes assessed as reduction in quisqualate-induced Ca2+ mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529965BDBM50529965(CHEMBL4441707)
Affinity DataIC50: 3.30nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in CHO-TREx cell membranes assessed as reduction in quisqualate-induced Ca2+ mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529973BDBM50529973(CHEMBL4513498)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529959BDBM50529959(CHEMBL4551786)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529959BDBM50529959(CHEMBL4551786)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529956BDBM50529956(CHEMBL4551238)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529956BDBM50529956(CHEMBL4551238)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529987BDBM50529987(CHEMBL4448788)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529987BDBM50529987(CHEMBL4448788)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529955BDBM50529955(CHEMBL4475143)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529974BDBM50529974(CHEMBL4544729)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529974BDBM50529974(CHEMBL4544729)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529955BDBM50529955(CHEMBL4475143)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529959BDBM50529959(CHEMBL4551786)
Affinity DataIC50: 4.10nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in CHO-TREx cell membranes assessed as reduction in quisqualate-induced Ca2+ mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529959BDBM50529959(CHEMBL4551786)
Affinity DataIC50: 4.10nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in CHO-TREx cell membranes assessed as reduction in quisqualate-induced Ca2+ mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529992BDBM50529992(CHEMBL4548820)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529992BDBM50529992(CHEMBL4548820)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529993BDBM50529993(CHEMBL4548205)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529993BDBM50529993(CHEMBL4548205)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529954BDBM50529954(CHEMBL4446275)
Affinity DataIC50: 5.10nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in CHO-TREx cell membranes assessed as reduction in quisqualate-induced Ca2+ mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
Recordati

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529954BDBM50529954(CHEMBL4446275)
Affinity DataIC50: 5.10nMAssay Description:Negative allosteric modulation of human mGlu5 receptor expressed in CHO-TREx cell membranes assessed as reduction in quisqualate-induced Ca2+ mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
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