TargetNeutrophil elastase(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Inhibition of human Neutrophil elastaseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Inhibition of M2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human M3 receptorMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of PDE4B2 (unknown origin)More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of beta2 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of MMP12 (unknown origin)More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of MMP12 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG by high throughput automated patch clamp methodMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataEC50: 0.251nMAssay Description:Agonist activity at human beta2 adrenoceptorMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataEC50: 0.251nMAssay Description:Agonist activity at human beta2 adrenoceptorMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataEC50: 0.251nMAssay Description:Agonist activity at human beta2 adrenoceptorMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
School Of Pharmaceutical Sciences & The Fifth Affiliated Hospital
Curated by ChEMBL
Affinity DataEC50: 0.251nMAssay Description:Agonist activity at human beta2 adrenoceptorMore data for this Ligand-Target Pair