Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50010268
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50536995(CHEMBL4572971)
Affinity DataIC50:  8.81E+3nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50536988(CHEMBL4570691)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50536993(CHEMBL4517595)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50536994(CHEMBL4543045)
Affinity DataIC50:  2.39E+4nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50536992(CHEMBL4587347)
Affinity DataIC50:  2.49E+4nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50536991(CHEMBL4537434)
Affinity DataIC50:  3.32E+4nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50536987(CHEMBL4515491)
Affinity DataIC50:  6.33E+4nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50536989(CHEMBL4533068)
Affinity DataIC50:  1.07E+5nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50536990(CHEMBL4548885)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed