Affinity DataIC50: 0.0250nMAssay Description:Displacement of [125I]-(Glp1,Nle11,Try14)apelin-13 from recombinant rat EGFP-fused apelin receptor expressed in CHO cell membrane measured after 3 hr...More data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 568nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 176nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair