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Found 55 Enz. Inhib. hit(s) with all data for entry = 4930
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82562(CAS_182595 | NSC_182595 | S 14489)
Affinity DataKi:  0.610nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82518(CAS_124756-23-6 | MDL 73005 EF)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82563(CAS_182596 | NSC_182596 | S 15931)
Affinity DataKi:  1.51nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82367(CAS_141533-35-9 | SDZ 216,525 | SDZ 216-525)
Affinity DataKi:  1.58nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82564(CAS_132787 | NSC_132787 | S 15535)
Affinity DataKi:  1.77nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50026917(8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...)
Affinity DataKi:  1.99nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50280934(1-tert-Butylamino-3-(thiochroman-8-yloxy)-propan-2...)
Affinity DataKi:  8.31nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  9.33nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82369(CAS_133025-23-7 | WAY 100,135 | WAY 100135)
Affinity DataKi:  32.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82563(CAS_182596 | NSC_182596 | S 15931)
Affinity DataKi:  53.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  53.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM25764(ALPRENOLOL,(+) | ALPRENOLOL,(-) | Alfeprol | Alphe...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82563(CAS_182596 | NSC_182596 | S 15931)
Affinity DataKi:  115nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  115nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82562(CAS_182595 | NSC_182595 | S 14489)
Affinity DataKi:  141nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82562(CAS_182595 | NSC_182595 | S 14489)
Affinity DataKi:  151nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  170nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50280934(1-tert-Butylamino-3-(thiochroman-8-yloxy)-propan-2...)
Affinity DataKi:  182nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82563(CAS_182596 | NSC_182596 | S 15931)
Affinity DataKi:  191nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82564(CAS_132787 | NSC_132787 | S 15535)
Affinity DataKi:  214nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50026917(8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...)
Affinity DataKi:  234nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50280934(1-tert-Butylamino-3-(thiochroman-8-yloxy)-propan-2...)
Affinity DataKi:  363nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82562(CAS_182595 | NSC_182595 | S 14489)
Affinity DataKi:  372nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82563(CAS_182596 | NSC_182596 | S 15931)
Affinity DataKi:  417nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82518(CAS_124756-23-6 | MDL 73005 EF)
Affinity DataKi:  427nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82564(CAS_132787 | NSC_132787 | S 15535)
Affinity DataKi:  537nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82562(CAS_182595 | NSC_182595 | S 14489)
Affinity DataKi:  603nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  646nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  776nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  977nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82369(CAS_133025-23-7 | WAY 100,135 | WAY 100135)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50280934(1-tert-Butylamino-3-(thiochroman-8-yloxy)-propan-2...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82564(CAS_132787 | NSC_132787 | S 15535)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82518(CAS_124756-23-6 | MDL 73005 EF)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50026917(8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM25764(ALPRENOLOL,(+) | ALPRENOLOL,(-) | Alfeprol | Alphe...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  1.07E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  1.38E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50280934(1-tert-Butylamino-3-(thiochroman-8-yloxy)-propan-2...)
Affinity DataKi:  1.45E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82518(CAS_124756-23-6 | MDL 73005 EF)
Affinity DataKi:  1.62E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82564(CAS_132787 | NSC_132787 | S 15535)
Affinity DataKi:  1.74E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50026917(8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...)
Affinity DataKi:  1.74E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82369(CAS_133025-23-7 | WAY 100,135 | WAY 100135)
Affinity DataKi:  3.47E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM82369(CAS_133025-23-7 | WAY 100,135 | WAY 100135)
Affinity DataKi:  3.47E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM25764(ALPRENOLOL,(+) | ALPRENOLOL,(-) | Alfeprol | Alphe...)
Affinity DataKi:  4.47E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
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