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Found 47 Enz. Inhib. hit(s) with all data for entry = 50007358
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50:  7nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50:  7nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50:  14nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508783(CHEMBL3325515)
Affinity DataIC50:  16nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50:  18nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50:  21nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50:  26nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50:  28nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50:  29nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508787(CHEMBL3325519)
Affinity DataIC50:  34nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508781(CHEMBL4577391)
Affinity DataIC50:  36nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508782(CHEMBL3774725)
Affinity DataIC50:  39nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50:  49nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508784(CHEMBL4543868)
Affinity DataIC50:  50nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50:  51nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C double mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50:  52nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C double mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50:  55nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508789(CHEMBL3775346)
Affinity DataIC50:  60nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508792(CHEMBL4579182)
Affinity DataIC50:  63nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50:  73nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50:  74nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188H mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  105nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50:  107nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50:  111nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50:  126nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50:  126nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50:  166nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508781(CHEMBL4577391)
Affinity DataIC50: >200nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508781(CHEMBL4577391)
Affinity DataIC50: >200nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50:  236nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50:  293nMAssay Description:Inhibition of HIV1 reverse transcriptase V106M mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508791(CHEMBL4439382)
Affinity DataIC50:  303nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50:  377nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50:  415nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188H mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50:  468nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188H mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50:  494nMAssay Description:Inhibition of HIV1 reverse transcriptase V106M mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50:  630nMAssay Description:Inhibition of HIV1 reverse transcriptase V106M mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50:  798nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50:  894nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C double mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50:  926nMAssay Description:Inhibition of HIV1 reverse transcriptase V106M mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188H mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508786(CHEMBL4441079)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508788(CHEMBL4519998)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50:  2.76E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508780(CHEMBL4520231)
Affinity DataIC50:  3.88E+3nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508790(CHEMBL4584925)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508785(CHEMBL4459834)
Affinity DataIC50: >4.41E+4nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed