TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 2.40E+4nMAssay Description:Inhibition of recombinant full-length human N-terminal His6-tagged AKR1C3 expressed in Escherichia coli BL21 (DE3) using phenanthrenequinone as subst...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 1.53E+5nMAssay Description:Inhibition of recombinant full-length human N-terminal His6-tagged AKR1C3 expressed in Escherichia coli BL21 (DE3) using phenanthrenequinone as subst...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 measured after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 measured after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 measured after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 measured after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 measured after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 measured after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 125nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 132nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 156nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 233nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 measured after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 273nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using oracin as substrate measured after 30 mins in presence of NADPH ...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 326nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 measured after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataIC50: 348nMAssay Description:Inhibition of recombinant human AKR1C3 expressed in Escherichia coli BL21 (D3) using S-tetralol as substrate in presence of NADP+ by UV-spectrophotom...More data for this Ligand-Target Pair