Compile Data Set for Download or QSAR
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Found 31 Enz. Inhib. hit(s) with all data for entry = 50008902
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523410(CHEMBL4453475)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523415(CHEMBL4515188)
Affinity DataIC50:  4.74E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523412(CHEMBL4567098)
Affinity DataIC50:  7.56E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523409(CHEMBL4483725)
Affinity DataIC50:  8.54E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523406(CHEMBL4536433)
Affinity DataIC50:  8.95E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523408(CHEMBL4435264)
Affinity DataIC50:  9.41E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin IV [1-448](Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523411(CHEMBL4475207)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin IV [1-448](Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523410(CHEMBL4453475)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin IV [1-448](Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523409(CHEMBL4483725)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin IV [1-448](Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523406(CHEMBL4536433)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin IV [1-448](Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523408(CHEMBL4435264)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523408(CHEMBL4435264)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523411(CHEMBL4475207)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523409(CHEMBL4483725)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523411(CHEMBL4475207)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523408(CHEMBL4435264)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523412(CHEMBL4567098)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523410(CHEMBL4453475)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523415(CHEMBL4515188)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523412(CHEMBL4567098)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523410(CHEMBL4453475)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523406(CHEMBL4536433)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin IV [1-448](Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523415(CHEMBL4515188)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523409(CHEMBL4483725)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523406(CHEMBL4536433)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasmepsin IV [1-448](Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523412(CHEMBL4567098)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523415(CHEMBL4515188)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523411(CHEMBL4475207)
Affinity DataIC50:  2.17E+4nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523414(CHEMBL4436020)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523407(CHEMBL4438229)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523413(CHEMBL4576672)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed