TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 2.40E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 5.00E+4nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 510nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 810nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 2.80E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 4.10E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 3.10E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 6.40E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 6.00E+3nMAssay Description:Transactivation of GAL4-tagged human PPARgamma LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 210nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 2.60E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 6.50E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Transactivation of GAL4-tagged human PPARgamma LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 2.80E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 250nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 3.90E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
University Of Chieti "G. D.Annunzio
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair