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Found 11 Enz. Inhib. hit(s) with all data for entry = 50008828
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50522762(CHEMBL4475087)
Affinity DataIC50:  950nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50522755(CHEMBL4528755)
Affinity DataIC50:  1.82E+3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50522758(CHEMBL4473832)
Affinity DataIC50:  4.59E+3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50522753(CHEMBL4514758)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50522761(CHEMBL4465327)
Affinity DataIC50:  4.86E+3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50522754(CHEMBL4453336)
Affinity DataIC50:  5.88E+3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50522759(CHEMBL4461708)
Affinity DataIC50:  6.56E+3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50522757(CHEMBL4458937)
Affinity DataIC50:  8.84E+3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50522760(CHEMBL4471983)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
North China Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50522756(CHEMBL4532631)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged PARP1 expressed in Sf9 insect cells preincubated for 15 mins followed by NAD+ addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed