Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50007583
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510725(CHEMBL4560144)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510722(CHEMBL4572026)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510721(CHEMBL4568106)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510717(CHEMBL4446112)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510715(CHEMBL4544939)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510720(CHEMBL4476179)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50177729(Aplysamine-1 | aplysamine | CHEMBL380697)
Affinity DataKi:  30nMAssay Description:Inhibition of histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510726(CHEMBL4451014)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510714(CHEMBL4526393)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510719(CHEMBL4436457)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510724(CHEMBL4560119)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510718(CHEMBL4573388)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510723(CHEMBL4439125)
Affinity DataKi:  317nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510713(CHEMBL4476221)
Affinity DataKi:  374nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510716(CHEMBL4566980)
Affinity DataKi:  848nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK-293 cells incubated for 90 mins by radioligand displace...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510716(CHEMBL4566980)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510723(CHEMBL4439125)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510714(CHEMBL4526393)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510713(CHEMBL4476221)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510726(CHEMBL4451014)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510725(CHEMBL4560144)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510715(CHEMBL4544939)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510722(CHEMBL4572026)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510724(CHEMBL4560119)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510721(CHEMBL4568106)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510718(CHEMBL4573388)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510717(CHEMBL4446112)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510720(CHEMBL4476179)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Heinrich Heine University D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50510719(CHEMBL4436457)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed