Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50008162
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516324BDBM50516324(CHEMBL4457372)
Affinity DataIC50: 0.280nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516321BDBM50516321(CHEMBL4577209)
Affinity DataIC50: 0.290nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516308BDBM50516308(CHEMBL4469829)
Affinity DataIC50: 0.380nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516329BDBM50516329(CHEMBL4467363)
Affinity DataIC50: 0.570nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516307BDBM50516307(CHEMBL4445542)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes at -70 mV holding potential by two electrode voltage-clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516323BDBM50516323(CHEMBL4474129)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516337BDBM50516337(CHEMBL4594136)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516316BDBM50516316(CHEMBL4454928)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516325BDBM50516325(CHEMBL4463089)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516307BDBM50516307(CHEMBL4445542)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516322BDBM50516322(CHEMBL4447464)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 86240BDBM86240(Gly-L-Cys(1)-L-Cys(2)-L-Ser-L-Asn-L-Pro-L-Val-L-Cy...)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes by two electrode voltage-clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516343BDBM50516343(CHEMBL4535637)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516306BDBM50516306(CHEMBL4438403)
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516342BDBM50516342(CHEMBL4461998)
Affinity DataIC50: 6.40nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516314BDBM50516314(CHEMBL4462168)
Affinity DataIC50: 7.10nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516319BDBM50516319(CHEMBL4443205)
Affinity DataIC50: 7.70nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes by two electrode voltage-clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516309BDBM50516309(CHEMBL4594009)
Affinity DataIC50: 8.70nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516315BDBM50516315(CHEMBL4515208)
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516340BDBM50516340(CHEMBL4439678)
Affinity DataIC50: 9.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516331BDBM50516331(CHEMBL4583045)
Affinity DataIC50: 9.30nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516320BDBM50516320(CHEMBL4572578)
Affinity DataIC50: 9.80nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes by two electrode voltage-clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516313BDBM50516313(CHEMBL4459917)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516336BDBM50516336(CHEMBL4465982)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516339BDBM50516339(CHEMBL4461702)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516307BDBM50516307(CHEMBL4445542)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at rat alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding potentia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516311BDBM50516311(CHEMBL4516107)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516335BDBM50516335(CHEMBL4476528)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516325BDBM50516325(CHEMBL4463089)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at rat alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding potentia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445326BDBM50445326(CHEMBL3104239)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516310BDBM50516310(CHEMBL4470868)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516312BDBM50516312(CHEMBL4564474)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNicotinic acetylcholine receptor alpha9/alpha10(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445326BDBM50445326(CHEMBL3104239)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at rat alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516318BDBM50516318(CHEMBL4438463)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516308BDBM50516308(CHEMBL4469829)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at rat alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding potentia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516329BDBM50516329(CHEMBL4467363)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at rat alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding potentia...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516333BDBM50516333(CHEMBL4474223)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516332BDBM50516332(CHEMBL4461650)
Affinity DataIC50: 44nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516341BDBM50516341(CHEMBL4577266)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516338BDBM50516338(CHEMBL4458975)
Affinity DataIC50: 65nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516327BDBM50516327(CHEMBL4538537)
Affinity DataIC50: 77nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516330BDBM50516330(CHEMBL4454425)
Affinity DataIC50: 109nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516328BDBM50516328(CHEMBL4475498)
Affinity DataIC50: 115nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516317BDBM50516317(CHEMBL4457284)
Affinity DataIC50: 123nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445326BDBM50445326(CHEMBL3104239)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516334BDBM50516334(CHEMBL4582247)
Affinity DataIC50: 155nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516305BDBM50516305(CHEMBL4454376)
Affinity DataIC50: 161nMAssay Description:Antagonist activity at rat alpha3beta2 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516325BDBM50516325(CHEMBL4463089)
Affinity DataIC50: 168nMAssay Description:Antagonist activity at rat alpha3beta4 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516308BDBM50516308(CHEMBL4469829)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at rat alpha4beta2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
Veterans Affairs Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50516329BDBM50516329(CHEMBL4467363)
Affinity DataIC50: 341nMAssay Description:Antagonist activity at rat alpha3beta4 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
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