Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for entry = 50008861
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50522991(CHEMBL4473057)
Affinity DataIC50:  9.70nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) incubated for 30 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50522992(CHEMBL4444781)
Affinity DataIC50:  21nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) incubated for 30 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50522990(CHEMBL4476085)
Affinity DataIC50:  28nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) incubated for 30 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50522987(CHEMBL4460353)
Affinity DataIC50:  40nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) incubated for 30 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataIC50:  44nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) incubated for 30 mins by ELISAMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50522988(CHEMBL4462036)
Affinity DataIC50:  54nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) incubated for 30 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50522989(CHEMBL4468264)
Affinity DataIC50:  71nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) incubated for 30 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50522986(CHEMBL4443040)
Affinity DataIC50: >100nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) incubated for 30 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50522993(CHEMBL4464894)
Affinity DataIC50: >100nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) incubated for 30 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed