Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50009258
TargetSodium-dependent noradrenaline transporter(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50526691(CHEMBL4563913)
Affinity DataIC50: 8.20E+3nMAssay Description:Substrate activity at NET in human BE(2)-C cells assessed as inhibition of drug uptake by measuring MIBG IC50 incubated for 1 hr in presence of nonra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50526691(CHEMBL4563913)
Affinity DataIC50: 2.20E+4nMAssay Description:Substrate activity at NET in human SK-N-SH cells cells assessed as inhibition of drug uptake by measuring MIBG IC50 incubated for 1 hr in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50526691(CHEMBL4563913)
Affinity DataIC50: 2.39E+4nMAssay Description:Substrate activity at NET in human BE(2)-C cells cells assessed as inhibition of drug uptake by measuring MIBG IC50 incubated for 1 hr in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50526691(CHEMBL4563913)
Affinity DataIC50: 2.87E+4nMAssay Description:Substrate activity at NET in human BE(2)-C cells cells assessed as inhibition of drug uptake by measuring MIBG IC50 incubated for 1 hr in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50526691(CHEMBL4563913)
Affinity DataIC50: 3.52E+4nMAssay Description:Substrate activity at NET in human SK-N-SH cells cells assessed as inhibition of drug uptake by measuring MIBG IC50 incubated for 1 hr in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50526691(CHEMBL4563913)
Affinity DataIC50: 7.62E+4nMAssay Description:Substrate activity at NET in human SK-N-SH cells assessed as inhibition of drug uptake by measuring MIBG IC50 incubated for 1 hr in presence of nonra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed