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Found 29 Enz. Inhib. hit(s) with all data for entry = 50008750
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521844(CHEMBL4538158)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50305655(3-(6-(piperidin-1-yl)-9H-purin-2-yl)phenol | CHEMB...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521843(CHEMBL4457537)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521845(CHEMBL4451553)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521847(CHEMBL4460517)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521839(CHEMBL4581007)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521843(CHEMBL4457537)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521845(CHEMBL4451553)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50305655(3-(6-(piperidin-1-yl)-9H-purin-2-yl)phenol | CHEMB...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521842(CHEMBL4446836)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521846(CHEMBL4518384)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521843(CHEMBL4457537)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK-293-A2B cells incubated for 30 mins by scintillation counting method based radioli...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521842(CHEMBL4446836)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521843(CHEMBL4457537)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa-A2A cells incubated for 30 mins by scintillation counting method based radioli...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521844(CHEMBL4538158)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50305655(3-(6-(piperidin-1-yl)-9H-purin-2-yl)phenol | CHEMB...)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK-293-A2B cells incubated for 30 mins by scintillation counting method based radioli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521841(CHEMBL4468459)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521850(CHEMBL4438363)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521840(CHEMBL4442328)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50305655(3-(6-(piperidin-1-yl)-9H-purin-2-yl)phenol | CHEMB...)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa-A2A cells incubated for 30 mins by scintillation counting method based radioli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521849(CHEMBL4464139)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521839(CHEMBL4581007)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521841(CHEMBL4468459)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521847(CHEMBL4460517)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521848(CHEMBL4563248)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521838(CHEMBL4574873)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in HeLa-A3 cells incubated for 180 mins by scintillation counting method based radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521845(CHEMBL4451553)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK-293-A2B cells incubated for 30 mins by scintillation counting method based radioli...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521840(CHEMBL4442328)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO-A1 cells incubated for 60 mins by scintillation counting method based radioligand c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50521844(CHEMBL4538158)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa-A2A cells incubated for 30 mins by scintillation counting method based radioli...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed