Compile Data Set for Download or QSAR
maximum 50k data
Found 71 Enz. Inhib. hit(s) with all data for entry = 50008760
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521920(CHEMBL4469545)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521917(CHEMBL4520650)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521900(CHEMBL4580498)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521897(CHEMBL4567814)
Affinity DataKi:  0.980nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521905(CHEMBL4440527)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521892(CHEMBL4590762)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521921(CHEMBL4472410)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521896(CHEMBL4476077)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521898(CHEMBL4441517)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521909(CHEMBL4437469)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521922(CHEMBL4452479)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521913(CHEMBL4445108)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521899(CHEMBL4446721)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521915(CHEMBL4532772)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521890(CHEMBL4475996)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521895(CHEMBL4475337)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521906(CHEMBL4445915)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521916(CHEMBL4544209)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521901(CHEMBL4555424)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521904(CHEMBL4466325)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521903(CHEMBL4476491)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521910(CHEMBL4519332)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521910(CHEMBL4519332)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521908(CHEMBL4475060)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521912(CHEMBL4468164)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521914(CHEMBL4520766)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521902(CHEMBL4520830)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521893(CHEMBL4447876)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521907(CHEMBL4553438)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521920(CHEMBL4469545)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521894(CHEMBL4575677)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521891(CHEMBL4455631)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521919(CHEMBL4457031)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521899(CHEMBL4446721)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521905(CHEMBL4440527)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521903(CHEMBL4476491)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521904(CHEMBL4466325)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521890(CHEMBL4475996)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521916(CHEMBL4544209)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521918(CHEMBL4565876)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521893(CHEMBL4447876)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521901(CHEMBL4555424)
Affinity DataKi:  710nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521914(CHEMBL4520766)
Affinity DataKi:  740nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521911(CHEMBL4460203)
Affinity DataKi:  780nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521919(CHEMBL4457031)
Affinity DataKi:  830nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521895(CHEMBL4475337)
Affinity DataKi:  860nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521900(CHEMBL4580498)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521913(CHEMBL4445108)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521891(CHEMBL4455631)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50521909(CHEMBL4437469)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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